Drug Guide
415 drug entries: the why, not only the how much
Organized into 21 systems. Each entry explains the mechanism before the dose: that is what makes a regimen stick instead of being looked up every time.
Principles of Cardiovascular Regulation and Receptive Dynamics
Enalapril and Ramipril
Losartan and Valsartan
Sacubitril / Valsartan
Spironolactone and Eplerenone
Carvedilol and Metoprolol Succinate
Amlodipine and Nifedipine
Verapamil and Diltiazem
Furosemide
Hydrochlorothiazide and Chlorthalidone
Empagliflozin and Dapagliflozin
Acetylsalicylic Acid (Aspirin)
Clopidogrel and Ticagrelor
Rivaroxaban and Apixaban
Heparin Sodium and Enoxaparin
Amiodarone
Digoxin
Nitroglycerin and Sodium Nitroprusside
Integrated Summary of Clinical Adjustment and Safety
Bases of respiratory pharmacology
Salbutamol and Terbutaline
Salmeterol, Formoterol, Indacaterol, Olodaterol and Vilanterol
Ipratropium bromide
Tiotropium Bromide, Glycopyrronium, Aclidinium and Umeclidinium
Fluticasone, Budesonide, Beclomethasone and Ciclesonide
Prednisone, Methylprednisolone, Hydrocortisone and Dexamethasone
ICS/LABA, LAMA/LABA and Triple Therapy Associations (LAMA/LABA/ICS)
Theophylline and Aminophylline
Montelukast, Zafirlukast and Zileutón
Disodium Cromoglycate and Sodium Nedocromil
Omalizumab (Anti-IgE)
Biologicals Anti-IL5 (Mepolizumab, Reslizumab), Anti-IL5R$\alpha$ (Benralizumab) and Anti-IL4R$\alpha$ (Dupilumab)
Tezepelumab (Anti-TSLP)
N-Acetylcysteine, Erdocysteine, Dornase Alfa and Poractant Alfa
Codeine, Dextromethorphan, Cloperastine and Levodropropizine
Sildenafil, Bosentan, Ambrisentan, Epoprostenol and Riociguat
Nintedanib and Pirfenidone
Integration and Clinical Practice
Adrenaline (Epinephrine)
Norepinephrine (Norepinephrine)
Dopamine
Dobutamine
Phenylephrine
Clonidine
Salbutamol (Albuterol)
Propranolol
Metoprolol
Carvedilol
Labetalol
Tamsulosin
Phenoxybenzamine
Bethanechol
Pilocarpine
Neostigmine and Pyridostigmine
Donepezil
Atropine
Scopolamine (Hyoscine)
Ipratropium and Tiotropium Bromide
Oxybutynin
Succinylcholine (Suxamethonium)
Principles of Clinical Neuropharmacology
Fluoxetine
Venlafaxine
Amitriptyline
Mirtazapine
Selegiline
Haloperidol
Clozapine
Risperidone
Aripiprazole
Lithium Carbonate
Valproic Acid (Sodium Valproate)
Lamotrigine
Diazepam
Zolpidem
Methylphenidate
Donepezil
Synthesis and Comparative Tables
Physiopathological Bases and Dynamic Mechanisms of Action
Phenytoin
Carbamazepine
Oxcarbazepine
Ethosuximide
Phenobarbital
Gabapentin
Pregabalin
Vigabatrin
Topiramate
Levetiracetam
Brivaracetam
Lacosamide
Zonisamide
Perampanel
Levodopa / Carbidopa (and Benserazide)
Pramipexole
Ropinirole
Rotigotine
Entacapone / Tolcapone
Rasagiline
Safinamide
Biperiden
Amantadine
Synthesis and Comparative Tables of Advanced Pharmacotherapy
Bases of anesthetic pharmacology
Sevoflurane, Desflurane and Isoflurane
Nitrous Oxide and Xenon
Sodium Thiopental
Propofol
Etomidate
Ketamine
Dexmedetomidine and Clonidine
Fentanyl, Sufentanil and Remifentanil
Succinylcholine (Suxamethonium)
Cisatracurium, Rocuronium and Vecuronium
Sugammadex and Neostigmine
Procaine, Tetracaine and Benzocaine
Lidocaine, Bupivacaine and Ropivacaine
Ephedrine, Phenylephrine and Atropine
Dexamethasone, Ondansetron and Droperidol
Non-Opioid Strategies and Multimodal Blockade
Management Algorithms and Acute Crises
Comparative Table of the Anesthetic Vademecum
Physiopathological Bases of Pain and Inflammation
Paracetamol (Acetaminophen)
Metamizole (Dipyrone)
Ibuprofen
Ketorolac
Celecoxib
Morphine
Tramadol
Fentanyl
Sumatriptan
Methotrexate
Leflunomide
Adalimumab
Tofacitinib
Colchicine
Allopurinol
Synthesis: Atlas of Pharmacoselection and Toxicology
Principles of Hormonal Regulation and Therapeutic Adjustment
Metformin
Empagliflozin (and Dapagliflozin)
Liraglutide / Semaglutide
Sitagliptin
Glimepiride
Pioglitazone
Insulin Glargine and Insulin Lispro
Levothyroxine Sodium (T4)
Methimazole (Thiamazole) and Propyl hysteractyl (PTU)
Dexamethasone and Hydrocortisone
Fludrocortisone Acetate
Cabergoline and Octreotide
Desmopressin (DDAVP)
Alendronate Sodium and Zoledronic Acid
Denosumab and Teriparatide
Cinacalcet Hydrochloride
Atorvastatin (and Evolocumab)
Integrated Fit and Safety Summary
Dynamics of transporters in the nephron
Acetazolamide
Furosemide
Bumetanide
Torasemide
Ethacrynic Acid
Hydrochlorothiazide (HCTZ)
Chlorthalidone
Indapamide
Metolazone
Spironolactone
Eplerenone
Finerenone
Amiloride
Mannitol
Empagliflozin
Hopperptan
Cross-drug interactions of diuretics
Physiological Principles of Liquid Compartments
Physiology of Volume Regulation and Osmolarity
Isotonic Crystalloid Solutions
Hypotonic and Hypertonic Crystalloids
Colloid Solutions (Natural and Synthetic)
Sodium Disorders I: Hyponatremia
Sodium II Disorders: Hypernatremia
Potassium Disorders I: Hypokalemia
Potassium II Disorders: Hyperkalemia
Calcium Disorders
Magnesium Disorders
Phosphorus Disorders and Refeeding Syndrome Integration
Acid-Base Balance I: Classic Approach (Henderson-Hasselbalch)
Acid-Base Balance II: Physicochemical Approach (Stewart)
Metabolic Acidosis
Metabolic Alkalosis
Respiratory Disorders and Mixed Acid-Base Balance Disorders
Practical Prescription and Monitoring in Critical Patients
Integrated Summary of Solutions and Safe Infusion
Bases of gastrointestinal pharmacology
Omeprazole (and derivatives: Esomeprazole, Pantoprazole)
Famotidine
Sucralfate
Misoprostol
Aluminum Hydroxide, Magnesium Hydroxide and Calcium Carbonate
Metoclopramide
Domperidone and Cinitapride
Prucalopride and Linaclotide
Butylscopolamine and Trimebutine Hydroxide
Ondansetron
Aprepitant (and Fosaprepitant)
Lactulose, Macrogol (PEG) and Bisacodyl
Loperamide and Racecadotril
Mesalazine and Sulfasalazine
Azathioprine
Infliximab and Vedolizumab
Ursodeoxycholic Acid (UDCA), Pancreatin and Rifaximin
Synthesis and clinical application pearls
Introduction and Analysis Methodology
Unfractionated Heparin (UFH)
Enoxaparin Sodium (LMWH)
Fondaparinux Sodium
Warfarin Sodium / Acenocoumarol
Rivaroxaban / Apixaban
Dabigatran Etexilate
Acetylsalicylic acid (AAS)
Clopidogrel
Ticagrelor / Prasugrel
Glycoprotein IIb/IIIa Inhibitors (Abciximab / Tirofiban)
Alteplase (rt-PA) / Tenecteplase
Tranexamic Acid
Erythropoietic Agents (Epoetin Alfa / Darbepoetin)
Colony Stimulating Factors (Filgrastim / Pegfilgrastim)
Thrombopoietin analogues (Romiplostim / Eltrombopag)
Factor Replacement Therapies (Factor VIII / Factor IX)
Emicizumab
Idarucizumab / Andexanet Alfa
Deferasirox / Deferoxamine
Synthesis and Summary of Hematological Monitoring
Physiopathological Bases and Resistance Mechanisms
Benzylpenicillins and Isoxazolylpenicillins
Aminopenicillins and Beta-lactamase Inhibitors
First and Second Generation Cephalosporins
Third and Fourth Generation Cephalosporins
Fifth Generation Cephalosporins and Siderophores
Carbapenems
Monobactamics (Aztreonam)
Glycopeptides and Lipoglycopeptides
Aminoglycosides
Macrolides and Ketolides
Lincosamides (Clindamycin)
Tetracyclines and Glycylcyclines
Oxazolidinones
Cyclic Lipopeptides and Polymyxins
Fluoroquinolones
Sulfonamides and Cotrimoxazole
Nitroimidazoles (Metronidazole)
Fosfomycin and Nitrofurans
Azole Antifungals
Echinocandines and Historical Reserves
Synthesis: Integrated Antimicrobial Clinical Pathway
Biophysical mechanisms of pharmacological reversal
N-Acetylcysteine (NAC)
Atropine
Pralidoxime (2-PAM)
Flumazenil
Naloxone
Anti-Digoxin Antibody Fab Fragments
Fomepizole (4-Methylpyrazole)
Methylene Blue
Protamine Sulfate
Idarucizumab
Andexanet Alfa
Deferoxamine
Dimercaprol (BAL - British Anti-Lewisite)
Calcium Disodium Edetate (\(CaNa_2EDTA\))
Hydroxocobalamin (Vitamin B12a)
Physostigmine (Eserine)
Glucagon
Intravenous Lipid Emulsion (ILE - Intralipid)
Phytonadione (Vitamin K1)
Penicillamine (D-Penicillamine)
Summary of interactions and risks of antidotes
Key concepts in immunopharmacology, oncology and toxicology
Calcineurin inhibitors and immunophilias
Immunosuppressive antimetabolites
Monoclonal antibodies and anti-TNF therapies
Lymphocyte receptor and cytokine modulators
Alkylating agents and platinums
Antimetabolites and antitumor antibiotics
Inhibitors of microtubules and nuclear enzymes
Targeted oncological therapies (mAB and tyrosine kinase inhibitors)
Oncological hormone therapy and hormonal antagonists
Specific antidotes for drug poisoning
Chemical antidotes, environmental poisoning and chelators
New generation specific reverters
Analytical summary: systemic toxicities and their specific antidotes
Principles of Transepidermal Penetration and Vehicle Selection
Topical Retinoids: Tretinoin, Adapalene and Tazarotene
Systemic Retinoids: Isotretinoin and Acitretin
Topical Corticosteroids
Topical Calcineurin Inhibitors: Tacrolimus and Pimecrolimus
Methotrexate
Cyclosporin (Cyclosporin A)
Anti-TNF-α Biological Therapies: Adalimumab and Infliximab
Anti-IL-17 Biological Therapies: Secukinumab and Ixekizumab
Biological Therapies Anti-IL-12/23 (Ustekinumab) and Anti-IL-23 (Guselkumab, Risankizumab)
Dupilumab
Janus Kinase (JAK) Inhibitors: Tofacitinib, Ruxolitinib, Baricitinib and Abrocitinib
Antifungals: Terbinafine, Itraconazole and Fluconazole
Antimicrobials in Acne and Rosacea: Doxycycline, Minocycline and Topical Metronidazole
Antiparasitics: Ivermectin (Topical and Systemic) and Permethrin
Local and Systemic Oncological Therapies: Imiquimod, Topical 5-Fluorouracil and Vismodegib
Local Anesthetics: Lidocaine, Prilocaine and Bupivacaine
Integrated Summary of Pharmacological Adjustment and Safety
Physiology of Ocular Barriers and Topical Pharmacokinetics
Latanoprost, Travoprost, Bimatoprost
Timolol, Betaxolol
Brimonidine, Apraclonidine
Dorzolamide, Brinzolamide, Acetazolamide
Netarsudil
Pilocarpine
Atropine, Cyclopentolate, Tropicamide
Phenylephrine
Dexamethasone, Prednisolone, Fluorometholone, Loteprednol
Nepafenac, Ketorolac, Bromfenac
Olopatadine, Ketotifen, Alcaftadine
Ciclosporin A, Lifitegrast
Tobramycin, Moxifloxacin, Erythromycin
Ganciclovir, Acyclovir
Natamycin, Amphotericin B
Ranibizumab, Aflibercept, Faricimab, Bevacizumab
Fluorescein, Rose Bengal, Indocyanine Green
Hyaluronic Acid, Carboxymethylcellulose, Trehalose
Atlas of Pharmacological Selection and Systemic Toxicity Profile
Introduction and Gestational Pharmacokinetic Methodology
Oxytocin
Carbetocin
Misoprostol
Dinoprostone
Methylergometrine
Atosiban
Nifedipine
Beta-adrenergic (Ritodrine)
Magnesium sulfate
Indomethacin
Micronized Progesterone
Combined Oral Contraceptives (COCs)
Progestin-Only Contraceptives
Selective Estrogen Receptor Modulators (SERMs)
Aromatase Inhibitors
GnRH Modulators (Agonists and Antagonists)
Ovulation Inducers (Clomiphene Citrate / Gonadotropins)
Dopaminergic Agonists
Tranexamic Acid
Mifepristone and Methotrexate
Anti-D immunoglobulin
Maternal-Fetal Antimicrobials
Gestational Antihypertensives
Gestational Diabetes
Antenatal Corticosteroids
Synthesis and Summary of High Complexity Monitoring
Biochemical dynamics of micronutrients
Vitamin A (Retinol, Retinyl Esters and Carotenoids)
Vitamin D3 (Cholecalciferol) and Calcitriol
Vitamin E (Tocopherols and Tocotrienols)
Vitamin K (Phytonadione and Menaquinones)
Vitamin B1 (Thiamin)
Vitamin B2 (Riboflavin) and Vitamin B3 (Niacin)
Vitamin B5 (Pantothenic Acid) and Vitamin B6 (Pyridoxine)
Vitamin B7 (Biotin) and Vitamin B9 (Folic Acid)
Vitamin B12 (Cobalamin)
Vitamin C (Ascorbic Acid)
Calcium and Phosphorus
Iron (Load Physiology and Formulations)
Magnesium and Zinc
Trace elements: Selenium, Copper and Iodine
Omega-3 Polyunsaturated Fatty Acids (EPA and DHA)
Clinical Amino Acids: N-Acetylcysteine, Glutamine and Creatine
Probiotics and Prebiotics
Posological guidelines, limits and organic adjustment
Kinetic Principles of Systemic Oncological Treatment
Nitrogen Mustards and Oxazaphosphorines: Cyclophosphamide and Ifosfamide
Platinum Coordinates: Cisplatin, Carboplatin and Oxaliplatin
Pyrimidine Analogs: 5-Fluorouracil and Capecitabine
Folate Analogs at Oncogenic Doses: Methotrexate
Cytidine Analogues: Cytarabine and Gemcitabine
Anthracyclines and Intercalation Inhibitors: Doxorubicin and Epirubicin
Topoisomerase I and II inhibitors: Irinotecan and Etoposide
Microtubule Modulators (Taxanes): Paclitaxel and Docetaxel
Vinca Alkaloids: Vincristine and Vinblastine
Targeted Monoclonal Antibodies: Anti-HER2 (Trastuzumab and Pertuzumab)
Monoclonal Antibodies: Cetuximab (Anti-EGFR) and Bevacizumab (Anti-VEGF)
Selective Tyrosine Kinase Inhibitors: Imatinib and Osimertinib
Multikinase Inhibitors: Sorafenib and Regorafenib
Immune Checkpoint Inhibitors (Checkpoints): Pembrolizumab, Nivolumab and Ipilimumab
Oncological Endocrine Therapy: Tamoxifen, Anastrozole and Letrozole
CDK4/6 and PARP inhibitors: Palbociclib and Olaparib
Advanced Clinical Support: Febrile Neutropenia and Tumor Lysis Syndrome
Integrated Summary of Pharmacological Adjustment and Safety
Barrier Principles, Membrane Permeability and Topical Deposition
Ciprofloxacin / Dexamethasone (Otic)
Betahistine dihydrochloride
Methylprednisolone / Intratympanic Dexamethasone
Intratympanic Gentamicin
Fluticasone Propionate / Mometasone Furoate (Intranasal)
Bilastine / Rupatadine
Oxymetazoline Hydrochloride (Intranasal)
Montelukast Sodium
Nystatin / Fluconazole
Pilocarpine Hydrochloride
Benzydamine / Chlorhexidine (Mouthwashes and Sprays)
Amoxicillin/Clavulanic Acid
Ceftriaxone / Clindamycin (Systemic Use)
Methylprednisolone / Deflazacort
Adrenaline (Epinephrine) Nebulized
Tranexamic Acid
Topical Hemostatic Biomaterials
Integrated Summary of Adjustment, Pharmacokinetics and Safety
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